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Prostamax

Bioregulators

Also known as: Prostate Bioregulator, Prostamax Khavinson Peptide

Half-life: Short (minutes); biological effect persists via gene-expression modulation

Last reviewed:  ·  Published:

Anti AgingAnti Inflammatory

Overview

Prostamax is a short peptide bioregulator from the Khavinson family, designed for prostate health applications. It is proposed to target prostate epithelial gene expression to support normal prostate function, reduce inflammation in chronic prostatitis, and potentially modulate benign prostatic hyperplasia (BPH) progression. The compound is used in Russian clinical practice for chronic prostatitis, BPH, and as a general prostate-support measure in aging men.

Russian clinical-observational studies have reported improvements in IPSS (International Prostate Symptom Score), urinary flow measures, and inflammatory markers in patients with chronic prostatitis and BPH. The clinical evidence base is similar in character to that of other Khavinson bioregulators — predominantly Russian, predominantly observational, with limited Western validation.

Prostamax is sold by research-chemical vendors outside Russia. It should not be used as a substitute for proven BPH therapies (alpha-blockers, 5-alpha-reductase inhibitors) or as a substitute for proper urological evaluation in men with prostate symptoms, where ruling out malignancy is essential.

History

Prostamax was developed in the 2000s as part of the Khavinson bioregulator program for urological applications. The compound entered Russian clinical observational use in urology contexts through the 2000s and 2010s.

Effects

  • Reported improvement in chronic prostatitis symptoms
  • Possible reduction in BPH-related urinary symptoms
  • Anti-inflammatory effects in prostate tissue
  • Modulation of prostate gene expression
  • Russian observational support for elderly male prostate health

Side Effects

  • Generally well-tolerated in Russian clinical use
  • Mild injection-site reactions
  • Limited Western safety validation
  • Not a substitute for proper urological evaluation

Tolerability

Russian clinical use has reported good tolerability in urological patient populations. Western safety validation is essentially absent. Men with prostate symptoms should undergo proper urological evaluation (DRE, PSA, possibly imaging) before relying on any single agent for management — peptide bioregulators do not address the diagnostic question of whether symptoms represent BPH, chronic prostatitis, or malignancy.

Dosing Ranges

Prostate health support

Dose Range

1-5 mg

Frequency

Once daily (SubQ) or sublingual

Duration

10-20 day cycles, repeated 2-3 times per year

Dosing information is for educational purposes only. Consult a healthcare professional before using any peptide.

Reconstitution

Preparation Details

Typical Vial Size

20 mg

Water Type

Bacteriostatic water (BAC water)

Mixing Volume

2 mL

Half-Life

Short (minutes); biological effect persists via gene-expression modulation

Molecular Weight

~400-600 Da

Store reconstituted vial refrigerated at 2-8°C. Use within 21-30 days. Sublingual or subcutaneous administration is typical.

Calculate Prostamax dose

Regulatory Status

FDA Status

Not FDA approved.

Legal Status

Unregulated research chemical outside Russia.

USA

Not approved

Research-only

EU

Not approved

Not authorized as medicinal product

UK

Not approved

Classified as research chemical

Russia

Used in clinical practice

Used as bioregulator in Russian urology

Australia

Not approved

TGA has not evaluated

Canada

Not approved

Not authorized for human use

Cited Studies

Peptide regulation of aging: 35 years of research experience

Khavinson VK, Kuznik BI, Tarnovskaya SI, Linkova NS

Bulletin of Experimental Biology and Medicine (2015)

Foundational Khavinson-group review covering the full short-peptide bioregulator family including Prostamax.

View Study →

Mechanisms of biological action of short peptides: the role of cell genome regulation

Khavinson VK, Anisimov VN, Linkova NS, Bakhmet AA

Bulletin of Experimental Biology and Medicine (2020)

Modern Khavinson-group mechanistic review applicable to all tissue-targeting bioregulators including Prostamax.

View Study →

Peptide bioregulators in urological practice

Khavinson VK, Morozov VG, Anisimov VN

Advances in Gerontology (2016)

Russian-group review of peptide bioregulators in urological applications, providing observational support for Prostamax and related compounds in chronic prostatitis and BPH contexts.

View Study →

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