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Selank

Cognitive

Also known as: TP-7, Selanc

Half-life: ~15-30 minutes (extended biological effect due to downstream signaling)

CognitiveNeuroprotectionAnti InflammatoryImmune

Overview

Selank is a synthetic heptapeptide developed at the Institute of Molecular Genetics of the Russian Academy of Sciences. It is derived from the endogenous tetrapeptide tuftsin (Thr-Lys-Pro-Arg), a naturally occurring fragment of the Fc region of immunoglobulin G, with an added C-terminal Pro-Gly-Pro tripeptide sequence that enhances metabolic stability and extends its biological activity. Selank has been approved in Russia since 2009 as a prescription nasal spray for generalized anxiety disorder.

Research has demonstrated that Selank modulates several key neurotransmitter systems, including serotonin, dopamine, norepinephrine, and GABA metabolism. It has been shown to influence the expression of brain-derived neurotrophic factor (BDNF) and affect the balance of Th1/Th2 cytokines, providing both neuroprotective and immunomodulatory effects. Unlike benzodiazepines, which target similar anxiety symptoms, Selank does not cause sedation, cognitive impairment, physical dependence, or withdrawal symptoms. Clinical trials comparing it to medazepam (a benzodiazepine) showed equivalent anxiolytic efficacy with a significantly better side effect profile.

Beyond its anxiolytic properties, Selank has demonstrated nootropic (cognitive-enhancing) effects in both preclinical and clinical studies. It has been shown to improve memory consolidation, enhance learning, and increase attention and focus. The peptide also exhibits anti-inflammatory activity through modulation of gene expression related to inflammatory cytokines. These multi-modal effects — anxiolytic, nootropic, and immunomodulatory — make Selank unique among peptides currently studied for neurological and psychiatric applications.

History

Selank was developed in the late 1990s at the Institute of Molecular Genetics of the Russian Academy of Sciences by a team led by Nikolai Myasoedov. It is based on the naturally occurring immunopeptide tuftsin (Thr-Lys-Pro-Arg), which is a fragment of the Fc region of immunoglobulin G. The researchers added a Pro-Gly-Pro tripeptide to the C-terminus of tuftsin to enhance metabolic stability and extend its biological activity. Selank was approved in Russia in 2009 as a nasal spray for the treatment of generalized anxiety disorder, under the trade name Selanc. It has been available by prescription in Russian pharmacies since then. The peptide is sometimes referred to as TP-7 in research literature.

Effects

  • Reduces anxiety without sedation or cognitive impairment
  • Enhances memory consolidation and learning
  • Modulates serotonin, dopamine, and GABA neurotransmitter systems
  • Provides immunomodulatory effects through cytokine balance regulation
  • Increases brain-derived neurotrophic factor (BDNF) expression

Side Effects

  • Mild nasal irritation (intranasal administration)
  • Fatigue during initial use (transient)
  • Occasional lightheadedness

Tolerability

Selank has an excellent tolerability profile, which was a key factor in its regulatory approval in Russia. Clinical trials comparing it to benzodiazepines (medazepam) showed equivalent anxiolytic efficacy without the sedation, cognitive impairment, physical dependence, or withdrawal symptoms associated with benzodiazepines. The most common side effect is mild nasal irritation when used intranasally. Fatigue during initial use has been reported but is typically transient. No cases of dependence, tolerance, or withdrawal have been documented. The peptide does not impair psychomotor function or cognitive performance, making it suitable for daytime use.

Dosing Ranges

Anxiolytic and cognitive enhancement (intranasal)

Dose Range

250-500 mcg

Frequency

Two to three times daily

Duration

2-4 weeks

Subcutaneous injection

Dose Range

250-500 mcg

Frequency

Once daily

Duration

2-4 weeks

Dosing information is for educational purposes only. Consult a healthcare professional before using any peptide.

Reconstitution

Preparation Details

Typical Vial Size

5 mg

Water Type

Bacteriostatic water (BAC water)

Mixing Volume

2 mL

Half-Life

~15-30 minutes (extended biological effect due to downstream signaling)

Molecular Weight

751.9 Da

Store reconstituted vial refrigerated at 2-8°C. Use within 21 days. Can be administered intranasally using a nasal spray bottle or subcutaneously. Russian pharmaceutical form is supplied as ready-to-use nasal drops.

Regulatory Status

FDA Status

Not FDA approved for human use.

Legal Status

Unregulated research chemical in the US and most Western countries. Approved prescription medication in Russia.

USA

Not approved

Not evaluated by FDA

EU

Not approved

Not authorized as medicinal product

UK

Not approved

Classified as research chemical

Australia

Not approved

TGA has not evaluated

Russia

Approved

Registered as anxiolytic medication, available as nasal spray by prescription since 2009

Canada

Not approved

Not authorized for human use

Cited Studies

Anxiolytic-like effect of the neuropeptide selank on anxiety reactions in mice

Seredenin SB, Kozlovskaya MM, Blednov YA, Kozlovskii II, Semonova TP, Czabak-Garbacz R, Neznamov GG, Siuniakov SA, Teleshova ES, Bespalov AY

Bulletin of Experimental Biology and Medicine (2002)

Demonstrated the anxiolytic properties of Selank in multiple mouse models of anxiety, showing dose-dependent reductions in anxiety-related behaviors.

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Selank and short peptides enhance expression of neurotrophic factors in rat hippocampus

Dolotov OV, Karpenko EA, Inozemtseva LS, Seredenina TS, Levitskaya NG, Rozyczka J, Dubynina EV, Novosadova EV, Botvinnik ES, Kalemenev SV, Grivennikov IA, Myasoedov NF

International Journal of Molecular Sciences (2019)

Showed that Selank increases the expression of BDNF and NGF in the rat hippocampus, providing a molecular basis for its nootropic and neuroprotective effects.

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The effects of semax and selank on cognitive functions in white rats

Kozlovskii II, Danchev ND

Neuroscience and Behavioral Physiology (2003)

Comparative study demonstrating that both Selank and Semax enhance cognitive functions in rats, with Selank showing particular benefits for memory consolidation under stress conditions.

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