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Cartalax

Bioregulators

Also known as: Cartilage Bioregulator, AED, Cartalax Khavinson Peptide

Half-life: Short (minutes); biological effect persists via gene-expression modulation

Last reviewed:  ·  Published:

HealingAnti Aging

Overview

Cartalax is a short peptide bioregulator from the Khavinson family, designed for cartilage and connective-tissue applications. Reported as a tripeptide (Ala-Glu-Asp, AED) in some Khavinson-group publications, it is presumed to target chondrocyte gene expression to support cartilage matrix synthesis, slow age-related cartilage degradation, and aid in connective-tissue repair. The compound has been studied in Russian clinical-observational settings for osteoarthritis, sports injury recovery, and age-related joint dysfunction.

Russian clinical reports have described improvements in joint pain, range of motion, and functional capacity in elderly osteoarthritis patients and in athletes recovering from cartilage injuries. The mechanism is presumed to involve restoration of more youthful chondrocyte gene expression patterns and increased synthesis of cartilage matrix components including type II collagen and proteoglycans.

Western clinical data on Cartalax specifically is essentially absent. The compound is sold by research-chemical vendors and used in self-experimentation for joint-support purposes. As with the broader Khavinson family, the Russian observational evidence base is real but lacks Western replication, and the compound should not replace evidence-based joint therapies in patients with significant osteoarthritis.

History

Cartalax was developed in the 2000s as part of the Khavinson group's tissue-specific bioregulator program. The cartilage-targeting member of the family was based on bioactive fractions of cartilage tissue extracts, with the active short-peptide sequence identified through fractionation and synthesis. The compound entered Russian clinical observational use in the 2000s and 2010s.

Effects

  • Reported support of chondrocyte function and cartilage matrix synthesis
  • Improvements in joint pain and mobility (Russian observational)
  • Possible slowing of age-related cartilage degradation
  • Recovery support after cartilage injury
  • Modulation of connective-tissue gene expression

Side Effects

  • Generally well-tolerated in Russian clinical use
  • Mild injection-site reactions
  • Limited Western safety validation

Tolerability

Russian clinical use has reported good tolerability across multiple study populations. Western safety validation is essentially absent. The compound has a small enough molecular footprint that systemic side effects are unlikely at typical doses, but as with all Khavinson bioregulators the absence of independent Western data limits how confidently the tolerability profile can be generalized.

Dosing Ranges

Joint / cartilage support

Dose Range

1-5 mg

Frequency

Once daily (SubQ) or sublingual

Duration

10-20 day cycles, repeated 2-3 times per year

Dosing information is for educational purposes only. Consult a healthcare professional before using any peptide.

Reconstitution

Preparation Details

Typical Vial Size

20 mg

Water Type

Bacteriostatic water (BAC water)

Mixing Volume

2 mL

Half-Life

Short (minutes); biological effect persists via gene-expression modulation

Molecular Weight

~333 Da (AED tripeptide)

Store reconstituted vial refrigerated at 2-8°C. Use within 21-30 days. Sublingual or subcutaneous administration is typical.

Calculate Cartalax dose

Regulatory Status

FDA Status

Not FDA approved.

Legal Status

Unregulated research chemical outside Russia.

USA

Not approved

Research-only

EU

Not approved

Not authorized as medicinal product

UK

Not approved

Classified as research chemical

Russia

Used in clinical practice

Used as bioregulator in Russian rheumatology and sports medicine

Australia

Not approved

TGA has not evaluated

Canada

Not approved

Not authorized for human use

Cited Studies

Peptide regulation of aging: 35 years of research experience

Khavinson VK, Kuznik BI, Tarnovskaya SI, Linkova NS

Bulletin of Experimental Biology and Medicine (2015)

Foundational Khavinson-group review covering the full short-peptide bioregulator family including Cartalax.

View Study →

Mechanisms of biological action of short peptides: the role of cell genome regulation

Khavinson VK, Anisimov VN, Linkova NS, Bakhmet AA

Bulletin of Experimental Biology and Medicine (2020)

Modern review of the gene-expression modulation mechanism proposed for all Khavinson bioregulators including Cartalax.

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Short peptides and cartilage homeostasis

Khavinson VK, Linkova NS, Trofimova SV

Advances in Gerontology (2018)

Russian-group review of short peptide bioregulators in cartilage homeostasis, providing the specific mechanistic and observational context for Cartalax.

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